平安! 发表于 2011-11-9 19:57
$ t0 u& T y8 v" o! G4 oPazopanib (100 mg/kg/day free base equivalent)
$ J: M6 C& |+ w9 u! Y. p: Y5 s 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
- o8 o/ P. U+ b. D$ u搜索了一下,原料一大堆。0 B( q* M, e5 |
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对不起!100mg/kg是用于移植瘤的,我弄错了。$ d6 Y* q% o# C$ Q
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以下是正版说明书的推荐用量。& i6 t* T9 w1 W3 O
2 `$ v( y# W6 j: C; r--------------------- DOSAGE AND ADMINISTRATION ----------------& q E' m; D! D/ S/ \) x
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
) j4 d4 {. K1 q, R( M- p3 `* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
9 a7 I' Y4 ]% G: f---------------------DOSAGE FORMS AND STRENGTHS --------------/ V. G& u' ^: x
200 mg tablets. (3) 6 D- z# t+ i; y+ O
-------------------------------CONTRAINDICATIONS------------------------ |